Internally Assess Inhibitors of Class IA and IB PI3K Isoforms Application Note
The InhibiScreen Kinase Inhibitor Assay is a phenotypically relevant testing model based on the suppression of in vitro basophil stimulation in whole blood treated with inhibitors of molecular targets such as PI3Kδ and PI3Kγ.
- Accelerate lead discovery and optimization phases of drug discovery
- Adaptable formats for both low and high throughput projects
- Specific cell-based assay for PI3K isoforms δ and γ
- Profile compounds in hours